Farestos

ACTIVE HALF-LIFE 6-7 Days
CLASSIFICATION Selective Estrogen Receptor Modulator
DOSAGE 10-40 mg/day
ACNE No
WATER RETENTION No
HBR No
HEPATOTOXICITY No
AROMATIZATION No
MANUFACTURER Pharmacom Labs - US
LAB TEST See Document
WAREHOUSE USA Warehouse 4
SUBSTANCE Toremifene Citrate ,

Farestos is a modern and advanced alternative to Clomid, effectively replacing all of its beneficial characteristics!

Toremifene Citrate is a selective estrogen receptor modulator (SERM) that originates from triphenylethylene. It was patented and received approval in Europe during the mid-1990s for the treatment of metastatic ER+ breast cancer in postmenopausal women.

In bodybuilding, men utilize toremifene citrate as a post-cycle therapy (PCT) medication to mitigate and/or inhibit the adverse effects of elevated estradiol due to the aromatization of various androgens used in cycles. Specifically, toremifene aids in restoring endogenous testosterone levels in the bloodstream and helps prevent estrogen-related side effects such as gynecomastia.

It is essential to note that toremifene citrate, as a SERM, functions as a genuine estrogen blocker, unlike aromatase inhibitors. Toremifene works by obstructing the action of estradiol at its receptor sites within various tissues. It achieves this by binding more effectively to these estradiol receptors than estradiol itself, occupying the space estradiol would typically bind to. Once bound, toremifene does not activate these receptors, preventing estradiol from attaching as they are already filled.

Toremifene does not reduce the overall levels of estradiol circulating in the bloodstream; it merely inhibits estradiol's action in specific tissues. This is the key distinction between it and aromatase inhibitors, which lower total estradiol levels in the bloodstream through their action on the aromatase enzyme that converts androgens into estradiol.

Chemically, toremifene is quite similar to tamoxifen, but it is a newer generation medication with fewer toxic side effects compared to tamoxifen.

However, there are some downsides associated with toremifene. Notably, it negatively impacts SHBG (Sex Hormone Binding Globulin) levels in the body. Clinical studies have shown that while toremifene does stimulate natural testosterone production, it also raises SHBG levels in the blood. Consequently, this may diminish cycle efficiency when taken during a cycle to address gynecomastia symptoms.

Additionally, regarding HPTA restoration and endogenous testosterone production in males, toremifene is less effective than tamoxifen at equivalent doses. Research has indicated that a daily dose of 60mg of toremifene increased testosterone levels in participants by 42%, which, although significant, is lower than the 71% increase observed with a standard 20mg daily dose of tamoxifen in the same study.

As a result, for a more effective increase in testosterone production, the recommended dosage of toremifene should reach up to 120mg per day. This dosage can be maintained for the first week of PCT, followed by 100mg per day in the second week, and then 60mg per day for the last 3-4 weeks of PCT. Of course, specific dosage should be tailored according to individual blood work findings.

There are no special requirements for taking toremifene. It can be taken before, during, or after meals and can be consumed in the morning or at night before sleeping. There is no need to divide the toremifene dosage throughout the day, as its half-life is about 5 days, allowing for stable blood levels to be maintained over a 24-hour period or longer without necessitating split doses.

The price listed is for one blister (50 pills). If you order a single blister, it will be shipped without the original box. To receive the original box, please order two blisters (100 pills).